European Journal of Chemistry

Synthesis and antimicrobial activity of some novel 2-azetidinones and 4-thiazolidinones derivatives

Article Sidebar

PDF
Published: Jun 30, 2013
DOI: https://doi.org/10.5155/eurjchem.4.2.98-101.714
Keywords:
Synthesis, 2-Azetidinones, 4-Thiazolidinones, Microwave technique, Antimicrobial activity, Halosubstituted Schiff bases
Section
Research Article
Issue
Vol. 4 No. 2 (2013): June 2013
Dates
Received 2012-12-02
Accepted 2013-01-08
Published 2013-06-30


Main Article Content

Shivaji Chavan
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
Sainath Zangade
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
Archana Vibhute
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India
Yeshwant Vibhute
Laboratory of Organic Synthesis, Department of Studies in Chemistry, Yeshwant Mahavidyalaya, Nanded-431602, India

Abstract

Several 2-azetidinones 2a-e and 4-thiazolidinones 3a-e have been synthesized from halo-substituted Schiff bases using conventional as well as microwave technique. The newly synthesized compounds were established on the basis of spectroscopic technique. Further, all compounds screened for antimicrobial activity against Bacillus subtilis, Escherichia coli, Aspergillus niger and Aspergillus flavus. Most of the titled compounds show potent activity.

4_2_98_101

icon graph This Abstract was viewed 2137 times | icon graph Article PDF downloaded 1219 times

How to Cite
(1)
Chavan, S.; Zangade, S.; Vibhute, A.; Vibhute, Y. Synthesis and Antimicrobial Activity of Some Novel 2-Azetidinones and 4-Thiazolidinones Derivatives. Eur. J. Chem. 2013, 4, 98-101.

Article Details

Share
Links for Article


Crossref - Scopus - Google - European PMC
Crossref
Scopus
Google Scholar
Europe PMC
References

[1]. Dave, T. K.; Purohit, D. H.; Akbari, J. D.; Joshi, S. H. Indian J. Chem. 2007, 46B, 352-356.

[2]. Patel, R. B.; Desai, P. S.; Desai, K. R.; Chikhalia, K. H. Indian J. Chem. 2006, 45B, 773-778.

[3]. Vijay, K. M. M. J.; Nagaraja, T. S.; Shameer, H.; Jayachandran, E.; Sreenivasa, G. M. J. Pharm. Sci. Res. 2009, 1, 83-92.

[4]. Udupi, R. H.; Kasinath, N.; Bhat, A. R. Indian J. Heterocycl. Chem. 1998, 17, 221-224.

[5]. Singh, G. S.; Mbukwa, E.; Pheko, T. Arkivoc 2007, 9, 80-90.

[6]. Chavan, A. A.; Pai, N. R. Molecules 2007, 12, 2467-2477.
http://dx.doi.org/10.3390/12112467
PMid:18065951

[7]. Havaldar, F. H.; Mishra, S. J. Indian J. Heterocycl. Chem. 2004, 13, 197-200.

[8]. Patel, K. H.; Metha, A. G. E-J. Chem. 2006, 3, 267-273.

[9]. Trautman, H. D.; Longe, L. M. J. Am. Chem. Soc. 1948, 70, 3436-3439.
http://dx.doi.org/10.1021/ja01190a064

[10]. Surray, A. R. J. Am. Chem. Soc. 1949, 71, 3354-3356.
http://dx.doi.org/10.1021/ja01178a023

[11]. French, G. Chem. Abstr. 1966, 65, 4439-4445.

[12]. Doran, W. J.; Sholen, H. A. J. Org. Chem. 1938, 3, 193-197.
http://dx.doi.org/10.1021/jo01220a001

[13]. Kuçukguzel, G.; Kocatepe, A.; De Clercq, E.; Sahin, F.; Gulluce, M. Eur. J. Med. Chem. 2006, 41, 353-359.
http://dx.doi.org/10.1016/j.ejmech.2005.11.005
PMid:16414150

[14]. Yadav, R.; Srivastav, S. D.; Srivastav, S. K. Indian J. Chem. 2005, 44B, 1262-1266.

[15]. Oza, H.; Joshi, D. Parekh, H. Indian J. Chem. 1998, 37B, 822-824.

[16]. Saundane, A. R.; Yarlakatti, M.; Walmik, P.; Katkar, V. J. Chem. Sci. 2012, 124, 469-481.
http://dx.doi.org/10.1007/s12039-011-0180-6

[17]. Patel, R. B.; Desai, P. S.; Desai, K. R.; Chikhalia, K. H. Indian J. Chem. B 2006, 45, 773-778.

[18]. Solankee, A. N.; Patel, K. P.; Patel, R. B. Pelagia Res. Lib. 2012, 3, 117-122.

[19]. Bouzroura, S.; Bentarzi, Y.; Kaoua, R.; Nedjar-koli, B.; Poulain-Martini, S.; Dunach, E. Org. Commun. 2010, 3, 8-14.

[20]. Zangade, S. B.; Mokle, S. S.; Shinde, A. T.; Vibhute, Y. B. Green Chem. Lett. Rev. 2013, 6, 123-127.
http://dx.doi.org/10.1080/17518253.2012.713123

[21]. Zangade, S.; Shinde, A.; Patil, A.; Vibhute, Y. Eur. J. Chem. 2012, 3, 208-210.
http://dx.doi.org/10.5155/eurjchem.3.2.208-210.581

[22]. Karamunge, K. G.; Sayed, M. A.; Vibhute, A. Y.; Vibhute, Y. B. J. Indian. Chem. Soc. 2011, 88, 443-446.

[23]. Zangade, S.; Mokle, S.; Chavan, S.; Vibhute, Y. Orbital: Electronic J. Chem. 2011, 3, 144-149.

[24]. Zangade, S. B.; Shinde, A. T.; Vibhute, A. Y.; Vibhute, Y. B. Pak. J. Chem. 2012, 2(1), 18-23.

[25]. Chavan, S. B.; Zangade, S. B.; Vibhute, A. Y. Vibhute, Y. B. Research J. Pharm. Bio. Chem. Sci. 2012, 3, 262-269.

[26]. Bouzroura, S.; Bentarzi, Y.; Kaoua, R.; Nedjar-Kolli, B.; Poulain-Martini, S.; Dunach, E. Org. Commun. 2010, 3(1), 8-14.

[27]. Pawar, R. P.; Andurkar, N. M.; Vibhute, Y. B. J. Indian. Chem. Soc. 1999, 76, 271-272.

[28]. Shinde, A. T.; Zangade, S. B.; Chavan, S. B.; Vibhute, A. Y.; Nalwar, Y. S.; Vibhute, Y. B. Synth. Commun. 2010, 40, 3506-3513.
http://dx.doi.org/10.1080/00397910903457332

[29]. Varma, S. Green Chem. 1999, 1, 43-55.
http://dx.doi.org/10.1039/a808223e

[30]. Borah, R.; Kalita, D. J.; Sarma J. C. Indian J. Chem. B 2002, 41, 1032-1038.

Supporting Agencies

University Grant Commission (No. 38‐267/2009), New Delhi, India
Most read articles by the same author(s)
TrendMD

Dimensions - Altmetric - scite_ - PlumX

Downloads and views

Downloads

Download data is not yet available.

Metrics

Metrics Loading ...
License Terms

License Terms

by-nc

Copyright © 2024 by Authors. This work is published and licensed by Atlanta Publishing House LLC, Atlanta, GA, USA. The full terms of this license are available at https://www.eurjchem.com/index.php/eurjchem/terms and incorporate the Creative Commons Attribution-Non Commercial (CC BY NC) (International, v4.0) License (http://creativecommons.org/licenses/by-nc/4.0). By accessing the work, you hereby accept the Terms. This is an open access article distributed under the terms and conditions of the CC BY NC License, which permits unrestricted non-commercial use, distribution, and reproduction in any medium, provided the original work is properly cited without any further permission from Atlanta Publishing House LLC (European Journal of Chemistry). No use, distribution, or reproduction is permitted which does not comply with these terms. Permissions for commercial use of this work beyond the scope of the License (https://www.eurjchem.com/index.php/eurjchem/terms) are administered by Atlanta Publishing House LLC (European Journal of Chemistry).